11H-Indeno[1,2-b]quinoxalin-11-one 2-(4-Ethylbenzylidene)hydrazone

Bibliographic Details
Parent link:Molbank
Vol. 2021, iss. 4.— 2021.— [M1299, 7 p.]
Main Author: Kovrizhina A. R. Anastasia Ruslanovna
Corporate Author: Национальный исследовательский Томский политехнический университет Инженерная школа новых производственных технологий Научно-образовательный центр Н. М. Кижнера
Other Authors: Samorodova E. I. Elizaveta Innokentjevna, Khlebnikov A. I. Andrey Ivanovich
Summary:Title screen
11H-Indeno[1,2-b]quinoxaline derivatives present an important type of nitrogen-containing heterocyclic compound that are useful intermediate products in organic synthesis and have potential pharmaceutical applications. A new 11H-indeno[1,2-b]quinoxalin-11-one-2-(4-ethylbenzylidene)hydrazone (compound 3) was synthesized. Compound 3 is the first example of an azine derivative based on the 11H-indeno[1,2-b]quinoxaline system. The Z,E-isomerism of compound 3 was investigated by DFT calculations. Bioavailability was evaluated in silico using ADME predictions. According to the ADME results, compound 3 is potentially highly bioavailable and has potential to be used for the treatment of neuroinflammation and ischemia–reperfusion injury.
Language:English
Published: 2021
Subjects:
Online Access:https://doi.org/10.3390/M1299
Format: Electronic Book Chapter
KOHA link:https://koha.lib.tpu.ru/cgi-bin/koha/opac-detail.pl?biblionumber=666275