The development of cyclotron‑based radiopharmaceuticals: a comprehensive review of 64Cu and 123I‑radiolabeled urea‑based small molecule PSMA ligands; Journal of Radioanalytical and Nuclear Chemistry; Vol. 332
| Parent link: | Journal of Radioanalytical and Nuclear Chemistry.— .— New York: Springer Science+Business Media LLC. Vol. 332.— 2023.— P. 3523-3546 |
|---|---|
| Corporate Author: | Томский политехнический университет |
| Other Authors: | Khasnovo Lutfi Aditjya, Larkina M. S. Mariya Sergeevna, Garapatski A. A. Alexander Alexandrovich, Yusubov M. S. Mekhman Suleiman-Ogly (Suleimanovich) |
| Summary: | 64Cu and 123I are attracting attention in taking up their role in the development and practical use of PSMA-targeting radiopharmaceuticals. The development of urea-based small molecule PSMA ligands labeled 64Cu and 123I has been progressing
steadily with the challenge of obtaining optimal performance as PSMA-targeting radiopharmaceutical for prostate cancer. In
this review, the authors provide an overview of recent research projects and future directions for the production of cyclotronbased medical radioisotopes 64Cu and 123I, and their application in the development of urea-based small molecule PSMA ligands labeled 64Cu and 123I as radiopharmaceuticals for prostate cancer. Текстовый файл |
| Language: | English |
| Published: |
2023
|
| Subjects: | |
| Online Access: | https://doi.org/10.1007/s10967-023-09048-3 |
| Format: | Electronic Book Chapter |
| KOHA link: | https://koha.lib.tpu.ru/cgi-bin/koha/opac-detail.pl?biblionumber=672771 |
Similar Items
Synthesis and Preclinical Evaluation of Urea-Based Prostate-Specific Membrane Antigen-Targeted Conjugates Labeled with 177Lu; ACS Pharmacology & Translational Science; Vol. 7, iss. 5
Published: (2024)
Published: (2024)
Single-Photon Emission Computer Tomography Imaging of Prostate-Specific Membrane Antigen (PSMA) Expression in Prostate Cancer Patients Using a Novel Peptide-Based Probe [99mTc]Tc-BQ0413 with Picomolar Affinity to PSMA: A Phase I/II Clinical Study; ACS Pharmacology & Translational Science; Vol. 8, iss. 3
Published: (2025)
Published: (2025)
Heterodimeric Radiotracer Targeting PSMA and GRPR for Imaging of Prostate Cancer—Optimization of the Affinity towards PSMA by Linker Modification in Murine Model; Pharmaceutics; Vol. 12, iss. 7
Published: (2020)
Published: (2020)
Preclinical Evaluation of a Novel High-Affinity Radioligand [ 99mTc]Tc-BQ0413 Targeting Prostate-Specific Membrane Antigen (PSMA); International Journal of Molecular Sciences; Vol. 24 - iss.24
Published: (2023)
Published: (2023)
Cyclotron Production of Iodine-124; Russian Physics Journal; Vol. 62, iss. 12
by: Salodkin S. S. Stepan Sergeevich
Published: (2020)
by: Salodkin S. S. Stepan Sergeevich
Published: (2020)
Synthesis, 123I-Radiolabeling Optimization, and Initial Preclinical Evaluation of Novel Urea-Based PSMA Inhibitors with a Tributylstannyl Prosthetic Group in Their Structures; International Journal of Molecular Sciences; Vol. 24, iss. 15
Published: (2023)
Published: (2023)
Quantitative evaluation of heat dissipation of a tellurium dioxide target front cooling during deuterons irradiation; Technical Physics; Vol. 69, No. 2
by: Salodkin S. S. Stepan Sergeevich
Published: (2024)
by: Salodkin S. S. Stepan Sergeevich
Published: (2024)
Preclinical Evaluation of the Copper-64 Labeled GRPR-Antagonist RM26 in Comparison with the Cobalt-55 Labeled Counterpart for PET-Imaging of Prostate Cancer; Molecules; Vol. 25, iss. 24
Published: (2020)
Published: (2020)
Novel Chlorin with a HYNIC: Synthesis, 99mTc-Radiolabeling, and Initial Preclinical Evaluation; Molecules; Vol. 30, iss. 1
Published: (2025)
Published: (2025)
Cyclotron Production of 99Mo Radionuclide by Bombarding Zirconium Targets with Alpha Particle Beams; Russian Physics Journal; Vol. 62, iss. 4
Published: (2019)
Published: (2019)
Source for In Situ Positron Annihilation Spectroscopy of Thermal-And Hydrogen-Induced Defects Based on the Cu-64 Isotope; Materials; Vol. 14, iss. 21
Published: (2021)
Published: (2021)
In situ изучение эволюции дефектной структуры в процессе воздействия водорода на композиты на основе магния и углеродных нанотрубок; Перспективы развития фундаментальных наук; Т. 1 : Физика
by: Саядян А. К.
Published: (2023)
by: Саядян А. К.
Published: (2023)
Reduction of Negative Charge in Mercaptoacetyl-Based Chelators Influences the Biodistribution of Prostate-Specific Membrane Antigen-Targeting Pseudopeptides Labeled with Technetium-99m; ACS Pharmacology & Translational Science; Vol. 8, iss. 10
Published: (2025)
Published: (2025)
Development of an automated unit for extraction-chromatographic separation of the 99Mo/99m Tc generator couple; Radiochemistry; Vol. 56, iss. 2
Published: (2014)
Published: (2014)
Synthesis of Radioiodinated Compounds. Classical Approaches and Achievements of Recent Years; International Journal of Molecular Sciences; Vol. 23, iss. 22
Published: (2022)
Published: (2022)
Evaluation of the Functional Suitability of Carboxylate Chlorin e6 Derivatives for Use in Radionuclide Diagnostics; Pharmaceutics; Vol. 18, iss. 1
Published: (2026)
Published: (2026)
Investigating characteristics of neutrons from accelerator-driven compact source using novel target of compressed beryllium-powder; Nuclear Instruments and Methods in Physics Research Section A: Accelerators, Spectrometers, Detectors and Associated Equipment; Vol. 1053
Published: (2023)
Published: (2023)
Positron Annihilation Spectroscopy Complex for Structural Defect Analysis in Metal–Hydrogen Systems; Materials; Vol. 15, iss. 5
Published: (2022)
Published: (2022)
66Ga-PET-imaging of GRPR-expression in prostate cancer: production and characterization of [66Ga]Ga-NOTA-PEG2-RM26; Scientific Reports; Vol. 11, iss. 1
Published: (2021)
Published: (2021)
Two-dimensional open quantum system in dissipative bosonic heat bath, external magnetic field, and two time-dependent electric fields; Physical Review E; Vol. 109, iss. 4
by: Alpomishev E. Kh.
Published: (2024)
by: Alpomishev E. Kh.
Published: (2024)
Phase I Clinical Study with the GRPR-Antagonist [99mTc]Tc-DB8 for SPECT Imaging of Prostate Cancer: Does the Injected Peptide Mass Make a Difference?; Pharmaceutics; Vol. 17, iss. 10
Published: (2025)
Published: (2025)
Разработка модели малогабаритного экстрактора с саморегулируемым уровнем границы раздела фаз для разделения пары 99Мо/99MТс; Известия Томского политехнического университета [Известия ТПУ]; Т. 323, № 3 : Химия
Published: (2013)
Published: (2013)
Investigation of ceramics based on Cu-Sn powder, obtained by plasma dynamic method; Energy Fluxes and Radiation Effects (EFRE-2016)
Published: (2016)
Published: (2016)
Получение нового наноколлоидного радиофармпрепарата на основе оксида алюминия; Известия Томского политехнического университета [Известия ТПУ]; Т. 323, № 3 : Химия
Published: (2013)
Published: (2013)
Current outlook on radionuclide delivery systems: from design consideration to translation into clinics; Journal of Nanobiotechnology; Vol. 17, iss. 1
Published: (2020)
Published: (2020)
New Cytochrome P-450 Ligands Based on Urea Derivatives; Pharmaceutical Chemistry Journal; Vol. 39, iss. 1
Published: (2005)
Published: (2005)
The dependency of fast neutron flux and spectra on the collimation-field size and geometry for fast neutron therapy purposes; Radiation Effects and Defects in Solids; Vol. 176, iss. 9-10
by: Shehada A. Abdullah
Published: (2021)
by: Shehada A. Abdullah
Published: (2021)
Influence of SBRT fractionation on TCP and NTCP estimations for prostate cancer; Physica Medica; Vol. 62
Published: (2019)
Published: (2019)
Radioiodination of small molecule PSMA ligand; Научная инициатива иностранных студентов и аспирантов
by: Lutfi Aditya Hasnowo
Published: (2023)
by: Lutfi Aditya Hasnowo
Published: (2023)
Cross section of the 96Zr(α,n)99Mo reaction induced by α-particles beams on natZr targets; Applied Radiation and Isotopes; Vol. 166
Published: (2020)
Published: (2020)
Dosimetric and radiobiological comparison of simultaneous integrated boost and sequential boost of locally advanced cervical cancer; Physica Medica; Vol. 73
Published: (2020)
Published: (2020)
Superhard nanocrystalline Ti-Cu-N coatings deposited by vacuum arc evaporation of a sintered cathode; Surface and Coatings Technology; Vol. 207
Published: (2012)
Published: (2012)
Способ получения и изучение биологических свойств меченной йодом-123 производной аминоглюкозы; Бюллетень сибирской медицины; Т. 17, № 1
Published: (2018)
Published: (2018)
Лазер на парах бромида меди со стабилизацией температуры стенок активного объема; Известия Томского политехнического университета [Известия ТПУ]; Т. 315. № 4: Энергетика
Published: (2009)
Published: (2009)
Получение радиофармацевтического препарата на основе производного глюкозы, меченного йодом-123; Физико-технические проблемы в науке, промышленности и медицине
by: Семенов А. С. Алексей Сергеевич
Published: (2015)
by: Семенов А. С. Алексей Сергеевич
Published: (2015)
Доклинические исследования радиофармацевтического лекарственного препарата на основе меченных 123I рекомбинантных адресных молекул для радионуклидной диагностики онкологических заболеваний с гиперэкспрессией HER-2/NEU; Изотопы: технологии, материалы и применение
by: Семенов А. А.
Published: (2023)
by: Семенов А. А.
Published: (2023)
Самоорганизация структуры CuCr контактного материала вакуумных выключателей при электронно-лучевом воздействии; Известия Томского политехнического университета [Известия ТПУ]; Т. 324, № 2 : Математика и механика. Физика
Published: (2014)
Published: (2014)
Preclinical Evaluation of 99mTc-Labeled GRPR Antagonists maSSS/SES-PEG2-RM26 for Imaging of Prostate Cancer; Pharmaceutics; Vol. 13, iss. 2
Published: (2021)
Published: (2021)
Оптимизация синтеза радиофармацевтического препарата "{123}I, йодофен"; Физико-технические проблемы в науке, промышленности и медицине
Published: (2016)
Published: (2016)
Preclinical Evaluation of the GRPR-Targeting Antagonist RM26 Conjugated to the Albumin-Binding Domain for GRPR-Targeting Therapy of Cancer; Pharmaceutics; Vol. 12, iss. 10
Published: (2020)
Published: (2020)
Similar Items
-
Synthesis and Preclinical Evaluation of Urea-Based Prostate-Specific Membrane Antigen-Targeted Conjugates Labeled with 177Lu; ACS Pharmacology & Translational Science; Vol. 7, iss. 5
Published: (2024) -
Single-Photon Emission Computer Tomography Imaging of Prostate-Specific Membrane Antigen (PSMA) Expression in Prostate Cancer Patients Using a Novel Peptide-Based Probe [99mTc]Tc-BQ0413 with Picomolar Affinity to PSMA: A Phase I/II Clinical Study; ACS Pharmacology & Translational Science; Vol. 8, iss. 3
Published: (2025) -
Heterodimeric Radiotracer Targeting PSMA and GRPR for Imaging of Prostate Cancer—Optimization of the Affinity towards PSMA by Linker Modification in Murine Model; Pharmaceutics; Vol. 12, iss. 7
Published: (2020) -
Preclinical Evaluation of a Novel High-Affinity Radioligand [ 99mTc]Tc-BQ0413 Targeting Prostate-Specific Membrane Antigen (PSMA); International Journal of Molecular Sciences; Vol. 24 - iss.24
Published: (2023) -
Cyclotron Production of Iodine-124; Russian Physics Journal; Vol. 62, iss. 12
by: Salodkin S. S. Stepan Sergeevich
Published: (2020)