Scalable total synthesis of natural vanillin-derived glucoside ω-esters

Detalhes bibliográficos
Parent link:Carbohydrate Research
Vol. 522.— 2022.— [108683, 7 p.]
Autor Corporativo: Национальный исследовательский Томский политехнический университет Исследовательская школа химических и биомедицинских технологий Лаборатория "Химическая инженерия и молекулярный дизайн"
Outros Autores: Avetyan (Avetian) D. L. David Ludvigovich, Shatskiy A. Andrey, Karkas M. D. Markus, Stepanova E. V. Elena Vladimirovna
Resumo:Title screen
The first total synthesis of vanilloloside, calleryanin, and a series of naturally occurring ω-esters of vanilloloside was realized through direct glycosylation of vanillin-based aglycones or late-stage derivatization of vanilloloside. All aglycones and their fragments were synthesized from vanillin as the sole aromatic precursor. Subsequently, these intermediates were used to construct various vanillin-derived glucoside ω-esters using a mild acidic deacetylation as the key synthetic step, providing the final products in the total yields of 10-50% and general purity of >95%. Additionally, the first operationally simple and sustainable synthesis of litseafoloside B was realized on large scale, avoiding the use of toxic solvents and reagents, providing an attractive alternative to isolation of this and other similar compounds from plant sources.
Режим доступа: по договору с организацией-держателем ресурса
Idioma:inglês
Publicado em: 2022
Assuntos:
Acesso em linha:https://doi.org/10.1016/j.carres.2022.108683
Formato: Recurso Electrónico Capítulo de Livro
KOHA link:https://koha.lib.tpu.ru/cgi-bin/koha/opac-detail.pl?biblionumber=668680

MARC

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330 |a The first total synthesis of vanilloloside, calleryanin, and a series of naturally occurring ω-esters of vanilloloside was realized through direct glycosylation of vanillin-based aglycones or late-stage derivatization of vanilloloside. All aglycones and their fragments were synthesized from vanillin as the sole aromatic precursor. Subsequently, these intermediates were used to construct various vanillin-derived glucoside ω-esters using a mild acidic deacetylation as the key synthetic step, providing the final products in the total yields of 10-50% and general purity of >95%. Additionally, the first operationally simple and sustainable synthesis of litseafoloside B was realized on large scale, avoiding the use of toxic solvents and reagents, providing an attractive alternative to isolation of this and other similar compounds from plant sources. 
333 |a Режим доступа: по договору с организацией-держателем ресурса 
461 |t Carbohydrate Research 
463 |t Vol. 522  |v [108683, 7 p.]  |d 2022 
610 1 |a электронный ресурс 
610 1 |a труды учёных ТПУ 
610 1 |a total synthesis 
610 1 |a natural occurring 
610 1 |a glycosides 
610 1 |a vanilloloside 
610 1 |a calleryanin 
610 1 |a esters of glycosides 
610 1 |a plant metabolites 
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610 1 |a гликозиды 
610 1 |a сложные эфиры 
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701 1 |a Karkas  |b M. D.  |g Markus 
701 1 |a Stepanova  |b E. V.  |c chemist  |c Associate Professor of Tomsk Polytechnic University, Candidate of Chemical Sciences  |f 1988-  |g Elena Vladimirovna  |3 (RuTPU)RU\TPU\pers\34245  |9 17776 
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